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          8種常見抗體藥物偶聯(lián)物(ADC)的不良反應及注意事項
          發(fā)布時間:2021-04-07     作者:axc   分享到:

          抗體**偶聯(lián)物(antibody-drug conjugate,ADC)是一類通過連接頭將靶標特異性的單克隆抗體與細胞*性藥物偶聯(lián)起來的靶向生物藥物,以單克隆抗體為載體將小分子細胞**以靶向方式運輸至目標**細胞中。

          目前已有8種ADC藥物(表1)。

                                                     表1 ADC**

          image.png

          抗體-藥物偶聯(lián)物(ADC產(chǎn)品目錄

          產(chǎn)品cas號產(chǎn)品名稱
          cas:159858-22-7Fmoc-Val-Cit-PAB
          cas:863971-53-3Fmoc-Val-Cit-PAB-PNP
          cas:55750-63-56-Maleimidohexanoic acid N-hydroxysuccinimide ester
          cas:159857-79-1Val-cit-PAB-OH
          cas:1116085-99-4Phe-Lys(Trt)-PAB
          cas:1116086-09-9Fmoc-Phe -Lys(Trt)-PAB-PNP
          cas:159857-79-1Val-Cit-PAB
          cas:253863-34-2Aloc-D-Ala-Phe-Lys(Aloc)-PAB-PNP
          cas:159857-90-6Cbz‐Phe‐(Alloc)Lys‐PAB‐PNP
          cas:1160844-44-9Boc‐Phe‐(Alloc)Lys‐PAB‐PNP
          cas:55750‐61‐3N-SMP
          cas:103750-03-45-Maleimidovalericacid-NHS
          cas:1325208-25-0Mal-PEG4-NHS
          cas:1260092-50-9Mal-PEG-NHS
          cas:756525-99-2Mal-PEG4-NHS-ester
          cas:1263044-56-9MC-PEG2-C2-NHS ester
          cas:132178-37-14-pentynoic acid succinimidyl ester
          cas:906564-59-85-hexynoic NHS ester
          cas:944251-24-5NHS-PEG4-azide
          cas:65869-64-9Bis-PEG1-NHS ester
          cas:65869-63-8Bis-PEG2-NHS Ester
          cas:1314378‐16‐9Bis-PEG3-NHS Ester
          cas:1314378-11-4NHS-PEG3-NHS
          cas:150244‐18‐1sulfo-LC-SPDP
          cas:1347750-84-8MAL-Tetra-EG-OPFP
          cas:1315355-92-0Mal-PEG5-NHS
          cas:1137109-21-7Mal-amido-PEG6-NHS
          cas:756525-93-6
          cas:1137109-22-8Mal-PEG10-NHS
          cas:824426-32-6Aeide-C1-NHS ester
          cas:1610796-02-5NHS-PEG12-azide
          cas:756526-03-1Bis-PEG5-NHS ester
          cas:1008402-79-6Bis-PEG9-NHS ester
          cas:870487-10-8Boc-Val-Cit-PAB-PNP
          cas:55683-37-9Propargyl-PEG1-acid
          cas:1174157-65-3Propargyl-PEG1-NHS ester
          cas:488150-84-1Propargyl-PEG1-Boc
          cas:3973-18-0Propynol Ethoxylate
          cas:203740-63-0Propargyl-PEG3-bromide
          cas:40842-04-4Bis-propargyl-PEG1
          cas:1835759-76-6Alkyne-PEG2-methylamine
          cas:1347750-80-4Alkyne-PEG4-thiol
          cas:1422540-81-5Alkyne-PEG4-5-nitrophenyl carbonate
          cas:89635-82-5Propargyl-PEG3-methane
          cas:1872433-63-0Alkyne-PEG4-(CH2)3-methyl ester
          cas:2183440-36-8APN-C3-PEG4-alkyne
          cas:52436-42-7Alkyne-PEG2-acrylate
          cas:2354291-37-3Gly-PEG3-endo-BCN, TFA salt
          cas:2110444-63-6Boc-Gly-PEG3-endo-BCN
          cas:15579-01-8Aminoethyl-SS-ethylalcohol
          cas:15579-00-7Aminoethyl-SS-propionic acid
          cas:51-85-4Aminoethyl-SS-ethylamine
          cas:485800-26-8t-Boc-Cystamine
          cas:2228857-32-5N3-SS-propionic acid
          cas:2144777-72-8N3-SS-PEG2-acid
          cas:2243566-44-9N3-SS-propionic NHS ester
          cas:1807540-82-4N3-SS-ethylalcohol
          cas:352305-38-5N3-SS-N3
          cas:1310827-27-0N3-PEG3-SS-PEG3-N3
          cas:2144777-83-1N3-PEG2-t-Butyl ester
          cas:1391914-41-2Alkyne-PEG1-SS-alcohol
          cas:1807503-85-0Alkyne-PEG1-SS-PEG1-acid
          cas:1817735-30-0Alkyne-PEG1-SS-PEG1-PFP ester
          cas:1964503-40-9Alkyne-PEG1-SS-PEG1-Alkyne
          cas:1807518-78-0Alkyne-PEG1-SS-PEG1-t-butyl ester
          cas:1807539-10-1Acid-PEG-SS-PEG-acid
          cas:485800-27-9Boc-NH-ethyl-SS-propionic acid
          cas:2128735-21-5Boc-aminooxy-ethyl-SS-propanol
          cas:864235-83-6Fmoc-NH-ethyl-SS-propionic acid
          cas:2128735-23-7Fmoc-NH-ethyl-SS-propionic NHS ester
          cas:2128735-24-8Mal-NH-ethyl-SS-propionic acid
          cas:5662-81-7Hydroxy-PEG3-SS-PEG3-alcohol
          cas:877864-04-5THP-SS-alcohol
          cas:1807503-88-3THP-SS-PEG1-t-butyl ester
          cas:1807512-37-3THP-SS-PEG1-Tos
          cas:1807530-16-02-hydroxyethyl disulfide mono-Tosylate
          cas:69981-39-1Bis-Tos-(2-hydroxyethyl disulfide)
          cas:1620523-64-9N3-SS-biotin
          cas:1430408-09-5DBCO-S-S-PEG3-biotin
          cas:142439-92-7Biotin-bisamido-SS-NHS
          cas:122266-55-1NHS-SS-biotin
          cas:325143-98-4Sulfo-NHS-SS-biotin
          cas:1869922-24-6PC Biotin-PEG3-alkyne
          cas:1937270-46-6PC Biotin-PEG3-N3
          cas:2353409-93-3PC Biotin-PEG3-NHS carbonate ester
          cas:1802907-98-7PC Alkyne-PEG4-NHS carbonate ester
          cas:1408057-91-9PC Methyltetrazine-PEG4-NHS carbonate ester
          cas:2353409-91-1PC N3-PEG11-NHS carbonate ester
          cas:2055041-38-6Mal-PEG2-Val-Cit-PAB-OH
          cas:Mal-PEG1-Val-Cit-PAB-PNP
          cas:2112738-13-1Mal-amido-PEG2-Val-Cit-PAB-PNP
          cas:2055024-65-0N3-PEG3-Val-Cit-PAB-OH
          cas:2055047-18-0N3-PEG3-Val-Cit-PAB-PNP
          cas:2353409-45-5BCN-PEG3-VC-PFP Ester
          cas:1367918-21-5Methylamino-PEG1-acid
          cas:1807521-03-4Methylamino-PEG1-Boc
          cas:1355197-57-7Methylamino-PEG-N3 (PEG1-PEGn)
          cas:85475-01-0Methylamino-PEG-Hydroxy (PEG1-PEGn)
          cas:2279944-69-1N,N'-DME-N-PEG2-tert-butyl ester
          cas:1817735-39-9N3-PEG2-sulfonic acid
          cas:255831-16-4Sulfonic acid-PEG3-sulfonic acid
          cas:112724-27-3Hydroxy-PEG2-C2-sulfonic acid
          cas:787524-78-1m-PEG4-sulfonic acid
          cas:1817735-29-7Sulfonic acid-PEG4-alkyne
          cas:1817735-32-2Boc-NH-PEG3-sulfonic acid
          cas:1817735-40-2Sulfonic acid-PEG2-t-Butoxycarbonyl
          cas:144942-89-2Amino-PEG-acid (PEG1-PEGn)
          cas:134978-97-5Amino-PEG-CH2COOH (PEG1-PEGn)
          cas:1263046-77-0Amino-PEG-(CH2)3COOH (PEG1-PEGn)
          cas:1260092-46-3Amino-PEG-t-butyl ester (PEG1-PEGn)
          cas:929-06-6Amino-PEG-alcohol (PEG1-PEGn)
          cas:2752-17-2Amino-PEG-Amine (PEG1-PEGn)
          cas:464190-91-8Amino-PEG-N3 (PEG1-PEGn)
          cas:1835759-88-0N3-PEG-methylamine (PEG1-PEGn)
          cas:1817735-43-5Amino-PEG-sulfonic acid (PEG1-PEGn)
          cas:2100306-60-1Amino-PEG-t-Boc-Hydrazide (PEG1-PEGn)
          cas:31576-51-9Amino-PEG-methyl (PEG1-PEGn)
          cas:122116-12-5Alkyne-PEG-amine (PEG1-PEGn)
          cas:1835759-76-6Propargyl-PEG2-methylamine
          cas:127828-22-2t-Boc-N-Amido-PEG-amine (PEG1-PEGn)
          cas:1351397-21-1Amino-PEG-benzyl ester (PEG1-PEGn)
          cas:1872433-72-1Trifluoroethyl-PEG-Amine (PEG1-PEGn)
          cas:2110448-97-8Gly-PEG-amine (PEG1-PEGn)
          cas:1020112-73-52-Amino-1,3-bis(carboxylethoxy)propane HCl salt
          cas:2055042-59-4N-(Amino-PEG3)-N-bis(PEG3-acid) HCl salt
          cas:2183440-35-7N-(acid-PEG3)-N-bis(PEG3-amine)
          cas:2183440-70-0N-(N3-PEG3)-N-(PEG2-amine)-PEG3-acid
          cas:174362-95-9Amino-Tri-(carboxyethoxymethyl)-methane
          cas:2100306-47-4N-(Amino-PEG1)-N-bis(PEG2-alkyne) HCl salt
          cas:2055040-99-6N-(Mal-PEG6)-N-bis(PEG3-amine) TFA salt

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